A facile synthesis of novel herbicidal 1-phenyl-piperazine-2,6-diones.

نویسندگان

  • Bin Li
  • Dong Xiang
  • Chi-Tung Hsu
  • Zhen-Long Liu
  • Chao Wu
  • Hua-Zheng Yang
چکیده

Novel 1-phenyl-piperazine-2,6-diones were prepared by a new facile synthetic route using methyl N-substituted iminomonoacetate as starting material. The structures of these compounds were established by (1)H-NMR, (13)C-NMR and GC/MS. 2-(4-Chloro-5-cyclo-pentyl-oxy-2-fluorophenyl)-tetrahydro-2H-pyrido-[1,2-a]-pyrazine-1,3-(4H,6H)-dione displayed the greatest herbicidal activity.

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عنوان ژورنال:
  • Molecules

دوره 10 9  شماره 

صفحات  -

تاریخ انتشار 2005